an efficient, three-component synthesis of 3,4-di hydropyrimidin-2(1h)-ones using lacl3/clch2cooh as environmentally benign and green catalytic system

Authors

b. pouramiri

e. tavakolinejad kermany

h. khajesamani

h. khabazzadeh

abstract

an improved, simple, and facile synthesis of 3,4-dihydropyrimidin-2(1h)-ones by employing three-component, one-pot condensation reaction of β-keto ester, aromatic aldehydes, and urea or n-methylurea using lacl3/clch2cooh as an inexpensive and green chemistry catalyst system under solvent-free conditions described. compared with the classicalbiginelli reaction conditions, this method has the advantages of good to excellent yields (80-99%) and short reaction time.

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Journal title:
journal of sciences, islamic republic of iran

Publisher: university of tehran

ISSN 1016-1104

volume 25

issue 4 2014

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